SCHEMBL2002956

SCHEMBL2002956

Cc1ccc2c(c1)c(C(=O)c1cnc(-c3cccnc3)o1)c(Cl)n2Cc1ccc(Cl)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES2 Q9H7Z7 3/20 0.44
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
ALOX15 P16050 1/20 0.43
ALOX12 P18054 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
HSD17B10 Q99714 1/20 0.43
FAAH O00519 1/20 0.43
MEN1 O00255 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41
ALOX5AP P20292 2/20 0.39
ALOX5 P09917 1/20 0.39
HDAC6 Q9UBN7 3/20 0.39
HDAC1 Q13547 2/20 0.39
TBXAS1 P24557 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.38
CYP1A2 P05177 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2004973 0.93 PTGES2 (0.42) PTGES2KDM4EALDH1A1MAPTHPGD
SCHEMBL1996791 0.92 PTGES2 (0.38) PTGES2KDM4EALDH1A1MAPTHPGD
SCHEMBL2003126 0.91 MEN1 (0.44) PTGES2KDM4EALDH1A1HSD17B10FAAH
SCHEMBL2003239 0.90 PTGES2 (0.41) PTGES2KDM4EALDH1A1MAPTHPGD
SCHEMBL2001978 0.90 FAAH (0.45) PTGES2KDM4EALDH1A1MAPTHPGD
SCHEMBL2007848 0.89 PTGES2 (0.45) PTGES2KDM4EALDH1A1MAPTHPGD
SCHEMBL1998318 0.89 HDAC6 (0.44) PTGES2KDM4EALDH1A1MAPTHPGD
SCHEMBL2002482 0.89 ALDH1A1 (0.44) PTGES2KDM4EALDH1A1MAPTHPGD
SCHEMBL2002164 0.88 ALOX5AP (0.45) PTGES2KDM4EALDH1A1MAPTHPGD
SCHEMBL2000862 0.88 PTGES2 (0.43) PTGES2KDM4EALDH1A1MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed