SCHEMBL19984499

SCHEMBL19984499

COC(=O)c1ccc2c(c1C)NC(=O)c1ccncc1S2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.39
ALDH1A1 P00352 3/20 0.39
GLA P06280 3/20 0.39
GAA P10253 3/20 0.39
CCNC P24863 2/20 0.36
CDK8 P49336 2/20 0.36
CYP46A1 Q9Y6A2 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.35
TP53 P04637 1/20 0.35
POLB P06746 1/20 0.35
THRB P10828 1/20 0.35
BLM P54132 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
FGFR1 P11362 1/20 0.35
SRC P12931 1/20 0.35
FGFR2 P21802 1/20 0.35
FGFR4 P22455 1/20 0.35
FGFR3 P22607 1/20 0.35
HPGD P15428 1/20 0.34
CASP1 P29466 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19984564 0.87 KDM4C (0.37) KDM4EALDH1A1GAACCNCCDK8
SCHEMBL18666975 0.83 TP53 (0.49) KDM4EALDH1A1GAAL3MBTL1TP53
SCHEMBL19984498 0.80 ALDH1A1 (0.39) KDM4EALDH1A1GLAGAACCNC
SCHEMBL19984562 0.78 MAPT (0.34) ALDH1A1GAAL3MBTL1TP53BLM
SCHEMBL17085917 0.70 KMT2A (0.50) KDM4EALDH1A1GAAHPGDHTT
SCHEMBL17085855 0.69 L3MBTL1 (0.48) KDM4EALDH1A1GAAL3MBTL1TP53
SCHEMBL2921667 0.69 CES1 (0.53) KDM4EGLAGAACYP46A1L3MBTL1
SCHEMBL17086097 0.69 KCNK3 (0.43) TP53HTT
SCHEMBL17086219 0.68 TP53 (0.39) L3MBTL1TP53POLBTHRBBLM
SCHEMBL19984503 0.66 KDM4C (0.37) KDM4EALDH1A1CCNCCDK8L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018053157-A1 HEPATITIS B CORE PROTEIN MODULATORS ASSEMBLY BIOSCIENCES, INC. (US) 2018-03-22 WO disclosed