SCHEMBL19984502

SCHEMBL19984502

CC(C)c1cc2c(cn1)OCCNC2=O

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
FABP6 P51161 1/20 0.48
GSK3B P49841 1/20 0.38
NTRK1 P04629 10/20 0.37
JAK2 O60674 7/20 0.37
MAPKAPK2 P49137 1/20 0.36
ALPL P05186 3/20 0.35
JAK3 P52333 3/20 0.34
ALK Q9UM73 3/20 0.34
ROS1 P08922 2/20 0.34
JAK1 P23458 2/20 0.34
NTRK2 Q16620 2/20 0.34
PLK4 O00444 1/20 0.34
NTRK3 Q16288 1/20 0.34
BTK Q06187 1/20 0.34
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22131521 0.81 FABP6 (0.51) FABP6GSK3BNTRK1JAK2MAPKAPK2
SCHEMBL18237530 0.79 ALDH1A1 (0.46) KDM4E
SCHEMBL18237989 0.78 MAOB (0.41)
SCHEMBL18237836 0.76 ALDH1A1 (0.42) KDM4E
SCHEMBL18238060 0.75 PARP10 (0.47) KDM4E
SCHEMBL13392164 0.74 FABP6 (0.61) FABP6GSK3BNTRK1JAK2MAPKAPK2
SCHEMBL2669110 0.72 FABP6 (0.48) FABP6GSK3BNTRK1JAK2MAPKAPK2
SCHEMBL18237940 0.72 PARP10 (0.47) KDM4E
SCHEMBL13306173 0.71 PTGS1 (0.35) KDM4E
SCHEMBL22607395 0.71 CLK4 (0.38) GSK3BNTRK1JAK2NTRK2NTRK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180079727-A1 9-MEMBERED FUSED RING DERIVATIVE SHIONOGI & CO., LTD. (JP) 2018-03-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180079727-A1 9-MEMBERED FUSED RING DERIVATIVE ACSS2, AGTR2, ACSL3 FABP6 2548/4885GSK3B 2144/4885NTRK1 4251/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.