SCHEMBL19984852

SCHEMBL19984852

Cc1cc(CNCc2nnc(-c3cnccn3)o2)n(C)n1

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.37
NLRP3 Q96P20 1/20 0.36
TERT O14746 4/20 0.34
PIEZO1 Q92508 9/20 0.33
HSD17B10 Q99714 1/20 0.32
SLC8A1 P32418 1/20 0.31
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19981277 0.79 TDP1 (0.45) KDM4EMEN1ALDH1A1MAPTKMT2A
SCHEMBL19973940 0.74 MAPK1 (0.33) KDM4ENLRP3MEN1KMT2A
SCHEMBL19973939 0.74 MAPK1 (0.33) KDM4ENLRP3MEN1KMT2A
SCHEMBL26777790 0.67 KDM4E (0.48) KDM4ENLRP3TERTPIEZO1HSD17B10
SCHEMBL19984983 0.66 KDM4E (0.47) KDM4ETERTPIEZO1HSD17B10MEN1
SCHEMBL19984827 0.65 KDM4E (0.44) KDM4ENLRP3TERTPIEZO1HSD17B10
SCHEMBL15599488 0.64 KDM4E (0.50) KDM4ETERTPIEZO1HSD17B10MEN1
SCHEMBL19984805 0.62 NPY5R (0.37) KDM4ENLRP3TERTPIEZO1MEN1
SCHEMBL579479 0.61 KDM4E (0.47) KDM4ETERTPIEZO1HSD17B10MEN1
SCHEMBL2077294 0.61 SMN1; SMN2 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018051255-A1 CYCLIC SUBSTITUTED-1,3,4-OXADIAZOLE AND THIADIAZOLE COMPOUNDS AS IMMUNOMODULATORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2018-03-22 WO disclosed