SCHEMBL19984977

SCHEMBL19984977

COc1ccccc1-c1nnc(CNC(=O)c2ncnc3[nH]ccc23)o1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
APLNR P35414 4/20 0.44
PARP1 P09874 3/20 0.42
KMT2A Q03164 1/20 0.42
ALDH1A1 P00352 2/20 0.41
NPC1 O15118 1/20 0.41
THRB P10828 1/20 0.41
HPGD P15428 1/20 0.41
MAPK1 P28482 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
USP2 O75604 1/20 0.41
ANO1 Q5XXA6 1/20 0.40
ANO2 Q9NQ90 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19984973 0.79 CYP3A4 (0.46) CYP3A4CYP2C9
SCHEMBL19984789 0.75 APLNR (0.54) APLNRPARP1KMT2AALDH1A1HPGD
SCHEMBL19984976 0.73 APLNR (0.54) APLNRPARP1KMT2AHPGDMAPK1
SCHEMBL19984815 0.70 KMT2A (0.48) APLNRKMT2AALDH1A1NPC1THRB
SCHEMBL16495669 0.69 WNT3A (0.46) APLNRKMT2AALDH1A1
SCHEMBL3828361 0.67 PTK2 (0.57) KMT2AALDH1A1NPC1THRBHPGD
Trifluoroacetic Acid SCHEMBL3822807 0.67 KMT2A (0.49) KMT2AALDH1A1NPC1THRBHPGD
SCHEMBL5122070 0.67 NEK1 (0.45) PARP1
SCHEMBL31060717 0.67 KMT2A (0.54) KMT2AALDH1A1NPC1THRBHPGD
SCHEMBL14289643 0.66 JAK2 (0.41) ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018051255-A1 CYCLIC SUBSTITUTED-1,3,4-OXADIAZOLE AND THIADIAZOLE COMPOUNDS AS IMMUNOMODULATORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2018-03-22 WO disclosed