SCHEMBL19986445

SCHEMBL19986445

O=C(NCCNc1c(Cl)cncc1Cl)Nc1ccc(Cl)c(F)c1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
CNR1 P21554 6/20 0.45
NAMPT P43490 2/20 0.44
SLC2A1 P11166 1/20 0.44
LMNA P02545 4/20 0.43
MAPT P10636 2/20 0.43
ALOX15 P16050 1/20 0.43
HSD17B10 Q99714 1/20 0.43
RAB9A P51151 2/20 0.43
TP53 P04637 1/20 0.43
HTT P42858 1/20 0.43
MAPK1 P28482 2/20 0.42
NPC1 O15118 2/20 0.42
HPGD P15428 1/20 0.42
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19986669 0.93 MEN1 (0.48) MEN1KMT2ACNR1NAMPTSLC2A1
SCHEMBL19986563 0.93 MEN1 (0.53) MEN1KMT2ACNR1NAMPTSLC2A1
SCHEMBL19986553 0.90 KMT2A (0.63) MEN1KMT2ASLC2A1LMNAMAPT
SCHEMBL19986506 0.88 MEN1 (0.43) MEN1KMT2ACNR1NAMPTLMNA
SCHEMBL19986566 0.86 MEN1 (0.51) MEN1KMT2ACNR1NAMPTSLC2A1
SCHEMBL19986700 0.84 LMNA (0.53) MEN1KMT2ACNR1NAMPTLMNA
SCHEMBL19986502 0.83 KMT2A (0.60) MEN1KMT2ASLC2A1LMNAMAPT
SCHEMBL19986628 0.81 MEN1 (0.56) MEN1KMT2ALMNAMAPTRAB9A
SCHEMBL19986530 0.81 ALOX15 (0.58) MEN1KMT2ASLC2A1LMNAMAPT
SCHEMBL19986578 0.81 MEN1 (0.41) MEN1KMT2ACNR1NAMPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113429341-A Novel capsid protein assembly inhibitors 正大天晴药业集团股份有限公司 2021-09-24 CN disclosed
CN-109790123-B Novel capsid protein assembly inhibitors 正大天晴药业集团股份有限公司 2021-06-25 CN disclosed
WO-2018050110-A1 NOVEL CAPSID PROTEIN ASSEMBLY INHIBITOR 正大天晴药业集团股份有限公司 2018-03-22 WO disclosed