SCHEMBL19986515

SCHEMBL19986515

O=C(NCCNc1c(Cl)cncc1Cl)c1ccc(F)c(Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNQ3 O43525 1/20 0.47
KCNQ2 O43526 1/20 0.47
KCNE1 P15382 1/20 0.47
KCNQ1 P51787 1/20 0.47
HPGD P15428 2/20 0.46
POLB P06746 1/20 0.46
HTT P42858 1/20 0.46
KMT2A Q03164 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.42
MEN1 O00255 1/20 0.42
HDAC3 O15379 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
PDE4D Q08499 1/20 0.41
MAOB P27338 2/20 0.41
CYP1A2 P05177 1/20 0.41
TSHR P16473 1/20 0.41
NFKB1 P19838 1/20 0.41
TAS1R3 Q7RTX0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19986648 0.93 KMT2A (0.50) KCNQ3KCNQ2KCNE1KCNQ1HPGD
SCHEMBL19986553 0.80 KMT2A (0.63) HTTKMT2ASMN1; SMN2MEN1CYP1A2
SCHEMBL19835598 0.78 HPGD (0.73) KCNQ3KCNQ2KCNE1KCNQ1HPGD
SCHEMBL19986516 0.77 KDM4E (0.43) POLBKMT2ASMN1; SMN2MEN1HDAC1
SCHEMBL6361467 0.76 KMT2A (0.61) KCNQ3KCNQ2KCNE1KCNQ1HPGD
SCHEMBL19986563 0.75 MEN1 (0.53) HTTKMT2ASMN1; SMN2MEN1CYP1A2
SCHEMBL24386507 0.74 HPGD (0.51) KCNQ3KCNQ2KCNE1KCNQ1HPGD
SCHEMBL19986502 0.73 KMT2A (0.60) HTTKMT2ASMN1; SMN2MEN1CYP1A2
SCHEMBL532006 0.73 TAS1R3 (0.51) KCNQ3KCNQ2KCNE1KCNQ1HPGD
SCHEMBL19986445 0.72 MEN1 (0.50) HPGDHTTKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113429341-A Novel capsid protein assembly inhibitors 正大天晴药业集团股份有限公司 2021-09-24 CN disclosed
CN-109790123-B Novel capsid protein assembly inhibitors 正大天晴药业集团股份有限公司 2021-06-25 CN disclosed
WO-2018050110-A1 NOVEL CAPSID PROTEIN ASSEMBLY INHIBITOR 正大天晴药业集团股份有限公司 2018-03-22 WO disclosed