SCHEMBL19986538

SCHEMBL19986538

CC(C)(CNc1c(Cl)cncc1Cl)CNS(=O)(=O)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.60
ALDH1A1 P00352 3/20 0.45
RAB9A P51151 3/20 0.40
LMNA P02545 4/20 0.40
MEN1 O00255 2/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
HTT P42858 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
PLAU P00749 1/20 0.38
SLC12A2 P55011 1/20 0.38
SLC12A5 Q9H2X9 1/20 0.38
PIK3CD O00329 1/20 0.38
PIK3CA P42336 1/20 0.38
PIK3CB P42338 1/20 0.38
MTOR P42345 1/20 0.38
PIK3CG P48736 1/20 0.38
PIK3C3 Q8NEB9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19986473 0.90 KMT2A (0.48) KMT2AALDH1A1RAB9ALMNAMEN1
SCHEMBL19986725 0.81 KMT2A (0.46) KMT2AALDH1A1RAB9ALMNAMEN1
SCHEMBL19986657 0.79 CCR1 (0.43) KMT2AALDH1A1LMNAMEN1CYP3A4
SCHEMBL19986720 0.71 RAB9A (0.49) KMT2AALDH1A1RAB9ALMNAMEN1
SCHEMBL28588269 0.71 CA1 (0.40) KMT2ARAB9ALMNAMEN1CYP3A4
SCHEMBL19986468 0.71 MEN1 (0.44) KMT2AALDH1A1RAB9ALMNAMEN1
SCHEMBL19986534 0.70 ALDH1A1 (0.46) KMT2AALDH1A1MEN1CYP3A4CYP2C9
SCHEMBL19986706 0.68 HTR2A (0.44) KMT2AALDH1A1MEN1CYP3A4CYP2C9
SCHEMBL25382079 0.66 KMT2A (0.54) KMT2AALDH1A1RAB9ALMNAMEN1
SCHEMBL21960093 0.66 ALDH1A1 (0.54) KMT2AALDH1A1LMNACYP2C19HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113429341-A Novel capsid protein assembly inhibitors 正大天晴药业集团股份有限公司 2021-09-24 CN disclosed
CN-109790123-B Novel capsid protein assembly inhibitors 正大天晴药业集团股份有限公司 2021-06-25 CN disclosed
WO-2018050110-A1 NOVEL CAPSID PROTEIN ASSEMBLY INHIBITOR 正大天晴药业集团股份有限公司 2018-03-22 WO disclosed