SCHEMBL19986657

SCHEMBL19986657

O=S(=O)(NCCCNc1c(Cl)cncc1Cl)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.43
KMT2A Q03164 5/20 0.43
MEN1 O00255 4/20 0.43
MAPT P10636 2/20 0.43
PKM P14618 2/20 0.43
HTT P42858 2/20 0.43
CYP1A2 P05177 3/20 0.43
CYP3A4 P08684 3/20 0.43
CYP2D6 P10635 3/20 0.43
CYP2C9 P11712 3/20 0.43
CYP2C19 P33261 3/20 0.43
ALDH1A1 P00352 2/20 0.42
LMNA P02545 1/20 0.42
POLB P06746 2/20 0.42
TP53 P04637 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
HTR2A P28223 4/20 0.41
HTR7 P34969 4/20 0.41
HTR6 P50406 4/20 0.41
DRD2 P14416 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19986725 0.92 KMT2A (0.46) CCR1KMT2AMEN1MAPTPKM
SCHEMBL19986706 0.89 HTR2A (0.44) KMT2AMEN1MAPTPKMHTT
SCHEMBL19986534 0.81 ALDH1A1 (0.46) KMT2AMEN1MAPTPKMCYP1A2
SCHEMBL19986538 0.79 KMT2A (0.60) KMT2AMEN1MAPTHTTCYP1A2
SCHEMBL10781482 0.75 ALDH1A1 (0.57) CCR1KMT2AMEN1MAPTPKM
SCHEMBL5320613 0.72 KMT2A (0.51) CCR1KMT2AMEN1MAPTHTT
SCHEMBL10904392 0.71 ALDH1A1 (0.49) CCR1KMT2AMEN1PKMCYP1A2
SCHEMBL9870626 0.70 FABP4 (0.68) PKMALDH1A1LMNATBXAS1
SCHEMBL19986658 0.70 HAO1 (0.35) KMT2AHTTALDH1A1L3MBTL1
SCHEMBL19986530 0.69 ALOX15 (0.58) KMT2AMEN1MAPTHTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113429341-A Novel capsid protein assembly inhibitors 正大天晴药业集团股份有限公司 2021-09-24 CN disclosed
CN-109790123-B Novel capsid protein assembly inhibitors 正大天晴药业集团股份有限公司 2021-06-25 CN disclosed
WO-2018050110-A1 NOVEL CAPSID PROTEIN ASSEMBLY INHIBITOR 正大天晴药业集团股份有限公司 2018-03-22 WO disclosed