SCHEMBL19986706

SCHEMBL19986706

O=S(=O)(NCCCNc1c(Cl)cncc1Cl)c1ccc(F)c(Cl)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.44
HTR7 P34969 6/20 0.44
HTR6 P50406 6/20 0.44
DRD2 P14416 5/20 0.44
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
PKM P14618 2/20 0.43
MAPT P10636 1/20 0.43
HTT P42858 1/20 0.43
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
ALDH1A1 P00352 2/20 0.42
TP53 P04637 1/20 0.42
AGTR1 P30556 1/20 0.42
GRIN1 Q05586 1/20 0.42
GRIN2A Q12879 1/20 0.42
GRIN2B Q13224 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19986534 0.93 ALDH1A1 (0.46) HTR2AHTR7HTR6DRD2MEN1
SCHEMBL19986657 0.89 CCR1 (0.43) HTR2AHTR7HTR6DRD2MEN1
SCHEMBL19986725 0.81 KMT2A (0.46) MEN1KMT2APKMMAPTHTT
SCHEMBL19986473 0.80 KMT2A (0.48) MEN1KMT2APKMMAPTALDH1A1
SCHEMBL19986468 0.80 MEN1 (0.44) MEN1KMT2APKMMAPTALDH1A1
SCHEMBL26921786 0.76 CYP3A4 (0.56) HTR2AHTR7HTR6DRD2MEN1
SCHEMBL19986648 0.73 KMT2A (0.50) KMT2AHTT
SCHEMBL19986707 0.72 STK17A (0.35) HTTCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL19986502 0.71 KMT2A (0.60) MEN1KMT2AMAPTHTTCYP1A2
SCHEMBL28588269 0.71 CA1 (0.40) MEN1KMT2AHTTCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113429341-A Novel capsid protein assembly inhibitors 正大天晴药业集团股份有限公司 2021-09-24 CN disclosed
CN-109790123-B Novel capsid protein assembly inhibitors 正大天晴药业集团股份有限公司 2021-06-25 CN disclosed
WO-2018050110-A1 NOVEL CAPSID PROTEIN ASSEMBLY INHIBITOR 正大天晴药业集团股份有限公司 2018-03-22 WO disclosed