SCHEMBL19986603

SCHEMBL19986603

Cc1cc(NC(=O)NCC2(CNc3c(C)cncc3C)CCOCC2)ccc1F

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 8/20 0.42
PIK3CD O00329 1/20 0.39
CYP3A4 P08684 1/20 0.39
AKT1 P31749 1/20 0.39
PIK3CA P42336 1/20 0.39
PIK3CB P42338 1/20 0.39
PIK3CG P48736 1/20 0.39
KCNJ6 P48051 4/20 0.38
KCNJ5 P48544 4/20 0.38
KCNJ3 P48549 4/20 0.38
KDR P35968 1/20 0.38
BLM P54132 1/20 0.38
CYP2C9 P11712 1/20 0.38
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
GRM4 Q14833 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19986607 0.90 NAMPT (0.41) NAMPTKCNJ6KCNJ5KCNJ3KDR
SCHEMBL19986694 0.90 NAMPT (0.41) NAMPTKCNJ6KCNJ5KCNJ3KDR
SCHEMBL19986634 0.85 KMT2A (0.41) NAMPTKCNJ6KCNJ5KCNJ3KDR
SCHEMBL19986602 0.82 KMT2A (0.47) CYP3A4MEN1KMT2A
SCHEMBL19986554 0.79 MEN1 (0.47) NAMPTKCNJ6KCNJ5KCNJ3KDR
SCHEMBL19986713 0.78 KCNJ6 (0.39) NAMPTCYP3A4KCNJ6KCNJ5KCNJ3
SCHEMBL19986668 0.78 KCNJ6 (0.39) NAMPTCYP3A4KCNJ6KCNJ5KCNJ3
SCHEMBL19986646 0.73 ALDH1A1 (0.49) CYP3A4MEN1KMT2A
SCHEMBL19986461 0.73 ALDH1A1 (0.52) CYP3A4MEN1KMT2A
SCHEMBL19986564 0.72 NAMPT (0.52) NAMPTKCNJ6KCNJ5KCNJ3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018050110-A1 NOVEL CAPSID PROTEIN ASSEMBLY INHIBITOR 正大天晴药业集团股份有限公司 2018-03-22 WO disclosed