SCHEMBL19994149

SCHEMBL19994149

COc1ccc(C2CCN(Cc3ccccc3)CC2OC(N)=O)cc1

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.51
SLC18A3 Q16572 2/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
CHRM2 P08172 1/20 0.48
CHRM3 P20309 1/20 0.48
MCHR1 Q99705 1/20 0.48
CHRM4 P08173 1/20 0.48
ACHE P22303 2/20 0.48
FAAH O00519 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16874602 0.82 MEN1 (0.63) SIGMAR1SLC18A3MEN1KMT2AACHE
SCHEMBL6042122 0.82 MEN1 (0.63) SIGMAR1SLC18A3MEN1KMT2AACHE
SCHEMBL16874797 0.82 MEN1 (0.63) SIGMAR1SLC18A3MEN1KMT2AACHE
SCHEMBL3488099 0.81 BCHE (0.47) SIGMAR1MEN1KMT2ACHRM2CHRM3
SCHEMBL19972380 0.80 SIGMAR1 (0.57) SIGMAR1SLC18A3MEN1KMT2AMCHR1
SCHEMBL28667637 0.79 ACHE (0.49) SIGMAR1MCHR1ACHE
SCHEMBL28453656 0.79 ACHE (0.49) SIGMAR1MCHR1ACHE
Hydrochloric Acid SCHEMBL28649444 0.78 ACHE (0.48) SIGMAR1MCHR1ACHE
SCHEMBL6360566 0.76 SIGMAR1 (0.63) SIGMAR1MEN1KMT2ACHRM4ACHE
SCHEMBL6046424 0.76 REN (0.49) SIGMAR1MEN1KMT2AMCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3515902-A1 6-MEMBERED CYCLIC AMINES OR LACTAMES SUBSTITUTED WITH UREA AND PHENYL Grünenthal GmbH (DE) 2019-07-31 EP disclosed
WO-2018054549-A1 6-MEMBERED CYCLIC AMINES OR LACTAMES SUBSTITUTED WITH UREA AND PHENYL Grünenthal GmbH (DE) 2018-03-29 WO disclosed