SCHEMBL20002488

SCHEMBL20002488

O=C(CO)N1CCC(C(=O)N2CCC(S(=O)(=O)c3ccc(F)cc3)C2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 4/20 0.47
NR1I2 O75469 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.46
ALDH1A1 P00352 2/20 0.45
EPHX2 P34913 1/20 0.44
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43
MAPT P10636 1/20 0.43
PKM P14618 1/20 0.43
ALOX12 P18054 1/20 0.43
HTR2A P28223 3/20 0.43
HTR2C P28335 2/20 0.43
KCNH2 Q12809 2/20 0.43
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
KDM4E B2RXH2 1/20 0.41
USP2 O75604 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002251 0.86 RORC (0.52) RORCNR1I2L3MBTL1ALDH1A1CCR5
SCHEMBL20002254 0.86 L3MBTL1 (0.48) RORCNR1I2L3MBTL1ALDH1A1EPHX2
SCHEMBL20002381 0.85 L3MBTL1 (0.56) RORCNR1I2L3MBTL1ALDH1A1EPHX2
SCHEMBL20002434 0.85 L3MBTL1 (0.56) RORCNR1I2L3MBTL1ALDH1A1EPHX2
SCHEMBL20002498 0.84 RORC (0.49) RORCL3MBTL1EPHX2MAPTHTR2A
SCHEMBL20002731 0.83 L3MBTL1 (0.48) RORCNR1I2L3MBTL1ALDH1A1EPHX2
SCHEMBL20003057 0.83 RORC (0.50) RORCL3MBTL1ALDH1A1EPHX2CA12
SCHEMBL20002743 0.83 L3MBTL1 (0.48) RORCNR1I2L3MBTL1ALDH1A1EPHX2
SCHEMBL20002790 0.83 L3MBTL1 (0.46) RORCNR1I2L3MBTL1ALDH1A1EPHX2
SCHEMBL20002878 0.83 L3MBTL1 (0.46) RORCNR1I2L3MBTL1ALDH1A1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed