SCHEMBL20002743

SCHEMBL20002743

O=C(C1CCSCC1)N1CCC(S(=O)(=O)c2ccc(F)cc2)C1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.48
EPHX2 P34913 1/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43
HTR2A P28223 3/20 0.42
HTR2C P28335 2/20 0.42
KCNH2 Q12809 2/20 0.42
ALDH1A1 P00352 2/20 0.42
RORC P51449 7/20 0.40
NR1I2 O75469 2/20 0.40
MAPT P10636 1/20 0.40
KDM4E B2RXH2 1/20 0.40
USP2 O75604 1/20 0.40
GAA P10253 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
DRD2 P14416 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002381 0.88 L3MBTL1 (0.56) L3MBTL1EPHX2CA12CA1CA2
SCHEMBL20002434 0.88 L3MBTL1 (0.56) L3MBTL1EPHX2CA12CA1CA2
SCHEMBL20002498 0.86 RORC (0.49) L3MBTL1EPHX2HTR2AHTR2CKCNH2
SCHEMBL20002254 0.85 L3MBTL1 (0.48) L3MBTL1EPHX2CA12CA1CA2
SCHEMBL20003057 0.85 RORC (0.50) L3MBTL1EPHX2CA12CA1CA2
SCHEMBL20002251 0.85 RORC (0.52) L3MBTL1ALDH1A1RORCNR1I2
SCHEMBL20002731 0.85 L3MBTL1 (0.48) L3MBTL1EPHX2CA12CA1CA2
SCHEMBL20002684 0.84 L3MBTL1 (0.47) L3MBTL1EPHX2CA12CA1CA2
SCHEMBL20002488 0.83 RORC (0.47) L3MBTL1EPHX2CA12CA1CA2
SCHEMBL20002790 0.82 L3MBTL1 (0.46) L3MBTL1EPHX2CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed