SCHEMBL2000262

SCHEMBL2000262

O=C(c1nnc(-c2ccncc2)o1)c1c(C(F)(F)F)n(Cc2ccc(Cl)cc2)c2ccc(O)cc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 4/20 0.48
LMNA P02545 3/20 0.48
PKM P14618 3/20 0.38
HTT P42858 3/20 0.36
MAPT P10636 3/20 0.36
ALDH1A1 P00352 2/20 0.36
GAA P10253 2/20 0.36
USP2 O75604 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ALOX5 P09917 1/20 0.35
ALOX5AP P20292 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
SMPD1 P17405 1/20 0.34
ALOX15 P16050 1/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34
ABCB11 O95342 2/20 0.33
HSP90AA1 P07900 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2006431 0.94 MAPK1 (0.50) MAPK1LMNAPKMHTTMAPT
SCHEMBL2006137 0.92 MAPT (0.42) MAPK1LMNAPKMMAPTALDH1A1
SCHEMBL2006683 0.91 MAPK1 (0.47) MAPK1LMNAPKMHTTMAPT
SCHEMBL2003185 0.90 PTGES2 (0.41) MAPK1LMNAPKMMAPTALDH1A1
SCHEMBL2002445 0.90 LMNA (0.43) MAPK1LMNAPKMMAPTALDH1A1
SCHEMBL2002430 0.89 MAPK1 (0.46) MAPK1LMNAPKMMAPTALDH1A1
SCHEMBL2005876 0.89 LMNA (0.50) MAPK1LMNAPKMHTTMAPT
SCHEMBL2004494 0.89 MAPK1 (0.52) MAPK1LMNAPKMHTTMAPT
SCHEMBL2004892 0.89 LMNA (0.35) MAPK1LMNAPKMHTTMAPT
SCHEMBL2007666 0.87 MAPK1 (0.43) MAPK1LMNAPKMMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed