SCHEMBL2005876

SCHEMBL2005876

O=C(c1nnc(-c2ccncc2)o1)c1c(C(F)(F)F)n(Cc2ccc(Cl)cc2)c2ccccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.50
MAPK1 P28482 3/20 0.50
PKM P14618 1/20 0.44
FAAH O00519 1/20 0.39
CES1 P23141 1/20 0.39
ALDH1A1 P00352 4/20 0.39
KDM4E B2RXH2 2/20 0.39
MITF O75030 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.38
HIF1A Q16665 1/20 0.37
PTGES2 Q9H7Z7 1/20 0.37
USP2 O75604 3/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
POLB P06746 1/20 0.36
TUBB4A P04350 1/20 0.36
TUBB P07437 1/20 0.36
TUBA3C P0DPH7 1/20 0.36
TUBA1B P68363 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2006816 0.94 LMNA (0.42) LMNAMAPK1PKMALDH1A1KDM4E
SCHEMBL2006431 0.91 MAPK1 (0.50) LMNAMAPK1PKMFAAHCES1
SCHEMBL2009227 0.91 CYP1A2 (0.42) LMNAMAPK1FAAHCES1ALDH1A1
SCHEMBL2003530 0.89 MAPK1 (0.45) LMNAMAPK1PKMFAAHCES1
SCHEMBL2000262 0.89 MAPK1 (0.48) LMNAMAPK1PKMFAAHCES1
SCHEMBL2002147 0.88 ALDH1A1 (0.37) LMNAMAPK1ALDH1A1KDM4EMITF
SCHEMBL2006683 0.88 MAPK1 (0.47) LMNAMAPK1PKMFAAHKDM4E
SCHEMBL2002436 0.88 LMNA (0.55) LMNAMAPK1PKMFAAHCES1
SCHEMBL2004831 0.87 PTGES2 (0.38) LMNAMAPK1ALDH1A1KDM4EHIF1A
SCHEMBL2002954 0.87 LMNA (0.54) LMNAMAPK1PKMFAAHCES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed