SCHEMBL20002758

SCHEMBL20002758

CC(C)(O)c1cccc(F)c1COC(C)(C(F)(F)F)C(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RORC P51449 13/20 0.36
HSD11B1 P28845 1/20 0.31
PDK1 Q15118 1/20 0.31
PDK2 Q15119 1/20 0.31
PDK3 Q15120 1/20 0.31
PDK4 Q16654 1/20 0.31
NR3C2 P08235 3/20 0.31
NR3C1 P04150 2/20 0.31
GUCY1B2 O75343 1/20 0.30
GUCY1A2 P33402 1/20 0.30
GUCY1A1 Q02108 1/20 0.30
GUCY1B1 Q02153 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18799682 0.85 RORC (0.40) RORC
SCHEMBL16886258 0.85 RORC (0.35) RORCHSD11B1PDK1PDK2PDK3
SCHEMBL20003145 0.85 RORC (0.35) RORCHSD11B1PDK1PDK2PDK3
SCHEMBL16892227 0.81 SMN1; SMN2 (0.35) RORCNR3C2NR3C1
SCHEMBL20002774 0.80 ACHE (0.36) RORC
SCHEMBL16886260 0.79 RORC (0.39) RORC
SCHEMBL20002812 0.78 TAAR1 (0.46)
SCHEMBL20002194 0.77 KDM1A (0.39) RORCNR3C2NR3C1
SCHEMBL20001981 0.75 RORC (0.37) RORCPDK1PDK2PDK3PDK4
SCHEMBL18214991 0.72 RORC (0.40) RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed