SCHEMBL20002194

SCHEMBL20002194

COc1cccc(F)c1COC(C)(C(F)(F)F)C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.39
MAOA P21397 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
MAPK1 P28482 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
SLC6A3 Q01959 1/20 0.37
KCNH2 Q12809 1/20 0.37
NR3C2 P08235 4/20 0.36
NR3C1 P04150 3/20 0.36
RORC P51449 4/20 0.36
SYK P43405 1/20 0.36
NFE2L2 Q16236 1/20 0.36
NPC1 O15118 1/20 0.35
LMNA P02545 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
PGR P06401 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18799682 0.87 RORC (0.40) RORC
SCHEMBL16886261 0.85 KDM1A (0.38) KDM1AMAOASMN1; SMN2MAPK1L3MBTL1
SCHEMBL20002774 0.81 ACHE (0.36) RORCKMT2A
SCHEMBL16886260 0.80 RORC (0.39) RORC
SCHEMBL20002812 0.79 TAAR1 (0.46) SMN1; SMN2L3MBTL1TDP1MEN1KMT2A
SCHEMBL16892228 0.78 L3MBTL1 (0.46) KDM1AMAOASMN1; SMN2MAPK1L3MBTL1
SCHEMBL20002758 0.77 RORC (0.36) NR3C2NR3C1RORC
SCHEMBL20001981 0.76 RORC (0.37) NR3C2NR3C1RORCPGR
SCHEMBL10190860 0.75 KDM1A (0.43) KDM1AMAOASMN1; SMN2MAPK1L3MBTL1
SCHEMBL18214991 0.73 RORC (0.40) SMN1; SMN2RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed