SCHEMBL20002854

SCHEMBL20002854

O=CN1CCC(C(=O)N2CCC([S+]([O-])c3ccc(F)cc3)C2)CC1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RORC P51449 2/20 0.42
MAPT P10636 1/20 0.38
PKM P14618 1/20 0.38
ALOX12 P18054 1/20 0.38
CYP46A1 Q9Y6A2 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
HSD11B1 P28845 8/20 0.37
LMNA P02545 1/20 0.37
KMT2A Q03164 1/20 0.37
GAA P10253 2/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
KDM4E B2RXH2 1/20 0.36
USP2 O75604 1/20 0.36
ALDH1A1 P00352 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002664 0.86 TSHR (0.41) PKML3MBTL1HSD11B1LMNAKMT2A
SCHEMBL20002286 0.86 TACR1 (0.45) RORC
SCHEMBL20002564 0.86 NAMPT (0.41) CYP46A1L3MBTL1HSD11B1LMNAKMT2A
SCHEMBL20002706 0.86 HSD11B1 (0.47) RORCL3MBTL1HSD11B1KMT2AALDH1A1
SCHEMBL20002698 0.86 HSD11B1 (0.47) RORCL3MBTL1HSD11B1KMT2AALDH1A1
SCHEMBL20002685 0.85 HSD11B1 (0.41) RORCMAPTPKMALOX12CYP46A1
SCHEMBL20002751 0.85 NOTUM (0.42) RORCMAPTL3MBTL1
SCHEMBL20002400 0.84 TACR3 (0.42) RORCMAPTL3MBTL1HSD11B1KMT2A
SCHEMBL20002340 0.83 TACR3 (0.39) CYP46A1L3MBTL1ALDH1A1
SCHEMBL22662762 0.83 SLC6A9 (0.43) RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed