SCHEMBL20002921

SCHEMBL20002921

CC(=O)N1CCC(N)(C(=O)N2CCC(S(=O)(=O)c3ccc(F)cc3)C2)CC1

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RORC P51449 16/20 0.44
NR1I2 O75469 2/20 0.43
CCR5 P51681 1/20 0.43
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
GPR6 P46095 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002866 0.89 RORC (0.49) RORCGPR6
SCHEMBL20002497 0.88 RORC (0.44) RORCNR1I2CCR5CYP11B1CYP11B2
SCHEMBL20002880 0.84 RORC (0.46) RORCNR1I2CCR5CYP11B1CYP11B2
SCHEMBL20002922 0.84 RORC (0.46) RORCNR1I2CCR5CYP11B1CYP11B2
SCHEMBL20003053 0.82 CCR5 (0.46) RORCNR1I2CCR5CYP11B1CYP11B2
SCHEMBL20002321 0.82 CCR5 (0.46) RORCNR1I2CCR5CYP11B1CYP11B2
SCHEMBL20002251 0.81 RORC (0.52) RORCNR1I2CCR5CYP11B1CYP11B2
SCHEMBL20002406 0.78 RORC (0.42) RORCCCR5
SCHEMBL20002869 0.77 RORC (0.44) RORCCCR5
SCHEMBL14413535 0.77 EPHX2 (0.47) RORCCCR5GPR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed