SCHEMBL20002922

SCHEMBL20002922

CC(=O)NC1(C(=O)N2CCC(S(=O)(=O)c3ccc(F)cc3)C2)CCN(C(C)=O)CC1

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RORC P51449 15/20 0.46
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
NR1I2 O75469 1/20 0.41
GPR6 P46095 1/20 0.41
CCR5 P51681 1/20 0.41
EPHX2 P34913 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002460 0.89 RORC (0.55) RORCGPR6EPHX2
SCHEMBL20002497 0.85 RORC (0.44) RORCCYP11B1CYP11B2NR1I2GPR6
SCHEMBL20002921 0.84 RORC (0.44) RORCCYP11B1CYP11B2NR1I2GPR6
SCHEMBL20002880 0.82 RORC (0.46) RORCCYP11B1CYP11B2NR1I2GPR6
SCHEMBL20003053 0.79 CCR5 (0.46) RORCCYP11B1CYP11B2NR1I2GPR6
SCHEMBL20002321 0.79 CCR5 (0.46) RORCCYP11B1CYP11B2NR1I2GPR6
SCHEMBL20002251 0.78 RORC (0.52) RORCCYP11B1CYP11B2NR1I2CCR5
SCHEMBL20002406 0.75 RORC (0.42) RORCCCR5EPHX2
SCHEMBL20002866 0.75 RORC (0.49) RORCGPR6EPHX2
SCHEMBL20002828 0.74 RORC (0.54) RORCCYP11B1CYP11B2NR1I2GPR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed