SCHEMBL20002866

SCHEMBL20002866

NC1(C(=O)N2CCC(S(=O)(=O)c3ccc(F)cc3)C2)CCCC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 4/20 0.49
EPHX2 P34913 1/20 0.42
HTR2A P28223 7/20 0.41
HTR2C P28335 6/20 0.41
KCNH2 Q12809 6/20 0.41
DRD2 P14416 4/20 0.41
L3MBTL1 Q9Y468 1/20 0.39
MAPT P10636 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
ATM Q13315 1/20 0.38
GPR6 P46095 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002921 0.89 RORC (0.44) RORCGPR6
SCHEMBL14413535 0.81 EPHX2 (0.47) RORCEPHX2HTR2AHTR2CKCNH2
SCHEMBL20002489 0.80 RORC (0.46) RORCEPHX2HTR2AHTR2CKCNH2
SCHEMBL20002406 0.79 RORC (0.42) RORCEPHX2HTR2AHTR2CKCNH2
SCHEMBL20002869 0.79 RORC (0.44) RORCEPHX2HTR2AHTR2CKCNH2
SCHEMBL20002497 0.78 RORC (0.44) RORCGPR6
SCHEMBL13890294 0.78 EPHX2 (0.50) EPHX2HTR2AHTR2CKCNH2DRD2
SCHEMBL20002563 0.78 EPHX2 (0.45) EPHX2HTR2AHTR2CKCNH2DRD2
SCHEMBL20003153 0.77 RORC (0.41) RORCEPHX2HTR2AHTR2CKCNH2
SCHEMBL20002381 0.77 L3MBTL1 (0.56) RORCEPHX2L3MBTL1MAPTCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed