SCHEMBL2000328

SCHEMBL2000328

CCOc1ccc2c(c1)c(C(=O)c1ncc(-c3ccccc3)o1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 8/20 0.43
ALOX5 P09917 3/20 0.41
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
PLA2G2A P14555 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
NTRK1 P04629 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2001878 0.93 ALOX5AP (0.42) ALOX5APALOX5PTGS1PTGS2CYP3A4
SCHEMBL2004225 0.93 PLA2G2A (0.45) ALOX5APALOX5PTGS2PLA2G2ACYP3A4
SCHEMBL2002959 0.93 ALOX5AP (0.42) ALOX5APALOX5PTGS1PTGS2CYP3A4
SCHEMBL2006766 0.91 F2RL3 (0.40) ALOX5APCYP3A4CYP2C9NTRK1
SCHEMBL2002560 0.90 MAPT (0.40) ALOX5APCYP3A4
SCHEMBL2008081 0.90 FAAH (0.41) ALOX5APALOX5CYP3A4CYP2C9
SCHEMBL2008374 0.90 ALOX5AP (0.44) ALOX5APALOX5PTGS1PTGS2PLA2G2A
SCHEMBL2001077 0.89 PTGES2 (0.41) ALOX5AP
SCHEMBL1999580 0.88 MAPT (0.39) ALOX5APALOX5
SCHEMBL2004616 0.88 ALOX5AP (0.42) ALOX5APALOX5PTGS1PTGS2PLA2G2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed