SCHEMBL20003671

SCHEMBL20003671

O=Cc1c[nH]cc(-c2ccc(F)cc2)c1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.37
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 2/20 0.35
LMNA P02545 1/20 0.35
NR4A2 P43354 1/20 0.34
PTPN1 P18031 1/20 0.34
MAPT P10636 2/20 0.34
POLB P06746 1/20 0.34
AURKB Q96GD4 1/20 0.34
PIM1 P11309 2/20 0.33
CDC7 O00311 1/20 0.33
GSK3B P49841 1/20 0.33
HIPK2 Q9H2X6 1/20 0.33
CLK4 Q9HAZ1 1/20 0.33
ERCC1 P07992 1/20 0.33
ERCC4 Q92889 1/20 0.33
PIM3 Q86V86 1/20 0.33
BRD4 O60885 1/20 0.33
BCL2L1 Q07817 1/20 0.32
BAD Q92934 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18860850 0.83 CYP2A6 (0.37) ALDH1A1KDM4ELMNAPTPN1MAPT
SCHEMBL18031340 0.75 NR4A2 (0.40) NR4A2MAPTAURKBPIM1CDC7
SCHEMBL20351754 0.75 BRD4 (0.40) ALDH1A1NR4A2MAPTPIM1CDC7
SCHEMBL10396846 0.74 NR4A2 (0.47) PTGS1NR4A2MAPTPOLBERCC1
SCHEMBL22200868 0.73 ALDH1A1 (0.40) PTGS1ALDH1A1KDM4ELMNAPTPN1
SCHEMBL23158698 0.72 NR4A2 (0.38) PTGS1ALDH1A1KDM4ENR4A2AURKB
SCHEMBL14949020 0.72 MAPT (0.36) ALDH1A1NR4A2MAPTPOLBPIM1
SCHEMBL363193 0.72 KDM4E (0.46) ALDH1A1KDM4ELMNAAURKBBCL2L1
SCHEMBL17233734 0.71 AURKB (0.42) PTGS1ALDH1A1KDM4EPTPN1AURKB
SCHEMBL29757272 0.71 IKBKB (0.43) PTGS1AURKBPIM1CDC7GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299369-A1 PYRIDO-AZAHETERECYDIC COMPOUND AND PREPARATION METHOD AND USE THEREOF Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CN) 2018-03-28 EP disclosed