SCHEMBL20006965

SCHEMBL20006965

Cc1onc(-c2ccccc2)c1C(=O)Nc1ccc(C(C)C)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.75
MAPK1 P28482 1/20 0.72
SMN1; SMN2 Q16637 1/20 0.72
GHSR Q92847 1/20 0.68
PTGS2 P35354 1/20 0.66
TSHR P16473 2/20 0.65
MEN1 O00255 1/20 0.65
KMT2A Q03164 1/20 0.65
ALDH1A1 P00352 5/20 0.64
L3MBTL1 Q9Y468 2/20 0.64
ALOX12 P18054 1/20 0.64
KDM4E B2RXH2 1/20 0.64
HTT P42858 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12585052 0.87 MAPK1 (0.79) TP53MAPK1SMN1; SMN2GHSRPTGS2
SCHEMBL13501815 0.86 ALDH1A1 (0.84) TP53MAPK1SMN1; SMN2GHSRPTGS2
SCHEMBL20006970 0.86 TP53 (1.00) TP53MAPK1SMN1; SMN2GHSRPTGS2
SCHEMBL2841709 0.85 TP53 (0.65) TP53MAPK1SMN1; SMN2GHSRPTGS2
SCHEMBL20006962 0.84 TP53 (0.72) TP53MAPK1SMN1; SMN2GHSRTSHR
SCHEMBL20006969 0.83 MAPK1 (0.72) TP53MAPK1SMN1; SMN2GHSRPTGS2
SCHEMBL31610836 0.82 GAA (0.76) TP53ALDH1A1L3MBTL1KDM4E
SCHEMBL19995013 0.81 GHSR (1.00) TP53MAPK1SMN1; SMN2GHSRTSHR
SCHEMBL20006967 0.80 TP53 (0.74) TP53MAPK1SMN1; SMN2GHSRTSHR
SCHEMBL13501824 0.79 KMT2A (0.69) TP53MAPK1SMN1; SMN2TSHRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018055235-A1 ISOXAZOLE-AMIDES FOR TREATING CARDIAC DISEASES UNIVERSITY OF HELSINKI (FI) 2018-03-29 WO disclosed