SCHEMBL20006969

SCHEMBL20006969

Cc1onc(-c2ccccc2)c1C(=O)Nc1ccc(C(C)(C)C)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.72
SMN1; SMN2 Q16637 1/20 0.72
PTGS2 P35354 2/20 0.71
ALDH1A1 P00352 4/20 0.69
L3MBTL1 Q9Y468 2/20 0.69
TP53 P04637 1/20 0.68
GHSR Q92847 1/20 0.68
ALOX12 P18054 1/20 0.64
KDM4E B2RXH2 1/20 0.64
TSHR P16473 1/20 0.62
HTT P42858 1/20 0.62
HPGD P15428 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12585052 0.87 MAPK1 (0.79) MAPK1SMN1; SMN2PTGS2ALDH1A1L3MBTL1
SCHEMBL13501815 0.86 ALDH1A1 (0.84) MAPK1SMN1; SMN2PTGS2ALDH1A1L3MBTL1
SCHEMBL20006965 0.83 TP53 (0.75) MAPK1SMN1; SMN2PTGS2ALDH1A1L3MBTL1
SCHEMBL20006968 0.81 PTGS2 (0.74) MAPK1SMN1; SMN2PTGS2ALDH1A1L3MBTL1
SCHEMBL9871174 0.81 PTGS2 (0.62) MAPK1SMN1; SMN2PTGS2ALDH1A1L3MBTL1
SCHEMBL20006970 0.81 TP53 (1.00) MAPK1SMN1; SMN2PTGS2ALDH1A1L3MBTL1
SCHEMBL19995013 0.81 GHSR (1.00) MAPK1SMN1; SMN2ALDH1A1TP53GHSR
SCHEMBL20006967 0.80 TP53 (0.74) MAPK1SMN1; SMN2ALDH1A1L3MBTL1TP53
SCHEMBL20006962 0.79 TP53 (0.72) MAPK1SMN1; SMN2ALDH1A1L3MBTL1TP53
SCHEMBL13501814 0.79 ALDH1A1 (0.68) MAPK1SMN1; SMN2ALDH1A1L3MBTL1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018055235-A1 ISOXAZOLE-AMIDES FOR TREATING CARDIAC DISEASES UNIVERSITY OF HELSINKI (FI) 2018-03-29 WO disclosed