SCHEMBL20008451

SCHEMBL20008451

C/C=C\C(=C/NCC)c1cc(N)ccc1Cl

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.34
CYP3A4 P08684 2/20 0.33
TSHR P16473 1/20 0.33
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CHRM2 P08172 1/20 0.30
CHRM3 P20309 1/20 0.30
MAOA P21397 1/20 0.30
HTR2C P28335 1/20 0.30
CHRNA4 P43681 1/20 0.30
HTR3A P46098 1/20 0.30
KCNH2 Q12809 1/20 0.30
HRH3 Q9Y5N1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7224774 0.67 P2RX7 (0.57) P2RX7CYP3A4TSHRCA1CA2
SCHEMBL20008147 0.65 CASP1 (0.35) CYP3A4TSHR
SCHEMBL27574494 0.64 P2RX7 (0.43) P2RX7CYP3A4TSHRCA1CA2
SCHEMBL13664886 0.63 CYP3A4 (0.35) P2RX7CYP3A4TSHRCA1CA2
SCHEMBL20008521 0.62
SCHEMBL22174797 0.62 CYP19A1 (0.38) CYP3A4TSHRMAOA
SCHEMBL21587030 0.62 P2RX7 (0.48) P2RX7TSHRCHRM2CHRM3MAOA
SCHEMBL1099858 0.61 CYP3A4 (0.48) P2RX7CYP3A4TSHRCA1CA2
SCHEMBL13689798 0.61 CYP3A4 (0.48) P2RX7CYP3A4TSHRCA1CA2
SCHEMBL3786681 0.61 CYP3A4 (0.48) CYP3A4TSHRCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299367-A1 BIARYL AMIDE COMPOUNDS AS KINASE INHIBITORS Novartis AG (CH) 2018-03-28 EP disclosed