SCHEMBL20008147

SCHEMBL20008147

C=CN/C=C(\C=C/C)c1cc(N)ccc1C

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 2/20 0.35
TSHR P16473 1/20 0.35
ALDH1A1 P00352 1/20 0.34
CYP3A4 P08684 1/20 0.32
PDE10A Q9Y233 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20009422 0.85 MEN1 (0.33) TSHR
SCHEMBL20008548 0.83 TP53 (0.31)
SCHEMBL20008186 0.82
SCHEMBL20008523 0.71 LMNA (0.34) ALDH1A1
SCHEMBL26084626 0.71 CASP1 (0.37) CASP1TSHRALDH1A1CYP3A4PDE10A
SCHEMBL20009423 0.71 MEN1 (0.36) TSHR
SCHEMBL20008773 0.70 CASP1 (0.42) CASP1TSHRALDH1A1CYP3A4PDE10A
SCHEMBL20009099 0.69
SCHEMBL19061357 0.69 CASP1 (0.41) CASP1TSHRALDH1A1CYP3A4PDE10A
SCHEMBL20009414 0.69 MEN1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299367-A1 BIARYL AMIDE COMPOUNDS AS KINASE INHIBITORS Novartis AG (CH) 2018-03-28 EP disclosed