SCHEMBL2000979

SCHEMBL2000979

O=C(c1ncc(-c2ccncn2)o1)c1c(Cl)n(Cc2ccc(Cl)cc2)c2ccccc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 3/20 0.45
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 2/20 0.39
MEN1 O00255 1/20 0.39
USP2 O75604 1/20 0.39
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39
KMT2A Q03164 1/20 0.39
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
MAPK10 P53779 1/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
SCD O00767 1/20 0.35
SCD5 Q86SK9 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2003811 0.91 FAAH (0.41) FAAHALDH1A1KDM4EMEN1KMT2A
SCHEMBL2006361 0.90 FAAH (0.45) FAAHCES1
SCHEMBL2000914 0.89 FAAH (0.42) FAAHALDH1A1KDM4EMEN1USP2
SCHEMBL2003432 0.89 LMNA (0.41) FAAHALDH1A1MEN1LMNAPOLB
SCHEMBL2004890 0.89 FAAH (0.39) FAAHALDH1A1KDM4EMEN1LMNA
SCHEMBL2008226 0.88 ALDH1A1 (0.41) ALDH1A1KDM4EMEN1USP2LMNA
SCHEMBL2006615 0.88 FAAH (0.42) FAAHALDH1A1KDM4EMEN1KMT2A
SCHEMBL2004673 0.86 ALDH1A1 (0.39) ALDH1A1KDM4EMEN1USP2LMNA
SCHEMBL2002842 0.86 MEN1 (0.43) FAAHALDH1A1MEN1LMNAKMT2A
SCHEMBL2002258 0.85 LMNA (0.39) ALDH1A1KDM4EMEN1USP2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed