SCHEMBL20021077

SCHEMBL20021077

Cc1cc2c(ccc(=O)n2CCN2CCOCC2)c(-c2ccc(Cl)cc2)c1CC(=O)O

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 6/20 0.44
KDM4E B2RXH2 4/20 0.43
ALDH1A1 P00352 4/20 0.43
CNR1 P21554 2/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.40
MDM4 O15151 1/20 0.39
PTGS2 P35354 1/20 0.39
MAPT P10636 2/20 0.39
HSD17B10 Q99714 2/20 0.39
GAA P10253 1/20 0.39
ALOX15 P16050 1/20 0.39
KMT2A Q03164 1/20 0.39
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
TNKS2 Q9H2K2 1/20 0.38
ACHE P22303 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10284225 0.81 KDM4E (0.44) KDM4EALDH1A1PTGDR2PTGS2MAPT
SCHEMBL20021131 0.81 PTGDR2 (0.47) KDM4EALDH1A1PTGDR2PTGS2MAPT
SCHEMBL3315614 0.80 CYP3A4 (0.41) CNR2KDM4EALDH1A1CNR1MDM4
SCHEMBL15182598 0.78 ALDH1A1 (0.37) CNR2KDM4EALDH1A1CNR1MDM4
SCHEMBL3326729 0.76 ACHE (0.47) KDM4EALDH1A1MAPTHSD17B10KMT2A
SCHEMBL3303958 0.74 KMT2A (0.49) KDM4EALDH1A1PTGDR2HSD17B10GAA
SCHEMBL3346070 0.69 KDM4E (0.43) KDM4EALDH1A1PTGDR2PTGS2MAPT
SCHEMBL20021094 0.69 MEN1 (0.46) KDM4EALDH1A1PTGDR2MAPTGAA
SCHEMBL20021162 0.69 KDM4E (0.43) KDM4EALDH1A1PTGDR2PTGS2MAPT
SCHEMBL20021151 0.67 MEN1 (0.44) KDM4EALDH1A1PTGDR2GAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2588455-B1 2-QUINOLINYL-ACETIC ACID DERIVATIVES AS HIV ANTIVIRAL COMPOUNDS GILEAD SCIENCES INC (US) 2018-04-04 EP disclosed