SCHEMBL20021228

SCHEMBL20021228

C#CCCCCCC(C)(NC)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.44
CYP1A2 P05177 2/20 0.44
CYP2D6 P10635 2/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
HSD17B10 Q99714 1/20 0.44
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 1/20 0.42
HPGD P15428 1/20 0.42
ACLY P53396 1/20 0.33
NAALAD2 Q9Y3Q0 1/20 0.33
FFAR1 O14842 1/20 0.33
CPT2 P23786 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
ACACB O00763 1/20 0.33
ACACA Q13085 1/20 0.33
CYP3A4 P08684 3/20 0.32
USP2 O75604 2/20 0.32
ALOX5 P09917 1/20 0.32
PTGS1 P23219 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18492198 0.93 CYP1A2 (0.38) MAPTCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL20021202 0.93 CYP1A2 (0.38) MAPTCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL18773764 0.86 ALDH1A1 (0.42) MAPTCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL7741623 0.78 CES2 (0.41) HSD17B10ALDH1A1FFAR1TDP1MEN1
SCHEMBL1012264 0.77 MAPT (0.42) MAPTCYP1A2CYP2D6CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL15799742 0.77 CES2 (0.40) HSD17B10ALDH1A1FFAR1TDP1MEN1
Hydrochloric Acid SCHEMBL15799582 0.77 CES2 (0.40) HSD17B10ALDH1A1FFAR1TDP1MEN1
SCHEMBL602186 0.75 ARG1 (0.53) MAPTCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL600737 0.75 ARG1 (0.53) MAPTCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL600736 0.75 ARG1 (0.53) MAPTCYP1A2CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3301108-A1 TRIAZOLE MACROCYCLE SYSTEMS Aileron Therapeutics, Inc. (US) 2018-04-04 EP disclosed