SCHEMBL2002134

SCHEMBL2002134

O=C(c1ncc(-c2cccnc2)o1)c1c(C(F)(F)F)n(Cc2ccc(Cl)cc2)c2ccc(Cl)cc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES2 Q9H7Z7 2/20 0.42
MCHR1 Q99705 1/20 0.38
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
MAPT P10636 2/20 0.37
ALOX15 P16050 2/20 0.37
ALOX12 P18054 2/20 0.37
HSD17B10 Q99714 2/20 0.37
HPGD P15428 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
ALOX5 P09917 1/20 0.36
ALOX5AP P20292 1/20 0.36
FAAH O00519 1/20 0.36
GRIN1 Q05586 2/20 0.35
GRIN2B Q13224 2/20 0.35
TBXAS1 P24557 1/20 0.35
SRPK1 Q96SB4 1/20 0.35
MEN1 O00255 1/20 0.34
CYP3A4 P08684 1/20 0.34
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2008949 0.94 PTGES2 (0.41) PTGES2MCHR1KDM4EALDH1A1MAPT
SCHEMBL2005859 0.94 PTGES2 (0.44) PTGES2MCHR1KDM4EALDH1A1MAPT
SCHEMBL2006671 0.92 PTGES2 (0.40) PTGES2MCHR1KDM4EALDH1A1MAPT
SCHEMBL2004581 0.92 ALOX5AP (0.41) PTGES2ALDH1A1MAPTALOX5ALOX5AP
SCHEMBL2002560 0.91 MAPT (0.40) PTGES2MAPTALOX15ALOX12HSD17B10
SCHEMBL2000666 0.91 PTGES2 (0.35) PTGES2MCHR1KDM4EALDH1A1MAPT
SCHEMBL2002959 0.91 ALOX5AP (0.42) PTGES2KDM4EALDH1A1MAPTHPGD
SCHEMBL2004214 0.91 CCR9 (0.37) PTGES2MCHR1KDM4EMAPTALOX15
SCHEMBL2000331 0.89 PTGES2 (0.41) PTGES2KDM4EALDH1A1MAPTALOX15
SCHEMBL4389111 0.88 LMNA (0.37) PTGES2MCHR1KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed