SCHEMBL2000666

SCHEMBL2000666

O=C(c1ncc(-c2cccnc2)o1)c1c(C(F)(F)F)n(Cc2ccc(Cl)cc2Cl)c2ccc(Cl)cc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES2 Q9H7Z7 1/20 0.35
RET P07949 1/20 0.35
FAAH O00519 1/20 0.35
ALDH1A1 P00352 4/20 0.34
LMNA P02545 4/20 0.34
MAPT P10636 3/20 0.34
ALOX12 P18054 2/20 0.34
KDM4E B2RXH2 2/20 0.34
POLB P06746 1/20 0.34
PKM P14618 1/20 0.34
HPGD P15428 1/20 0.34
TBXAS1 P24557 1/20 0.34
EPHX2 P34913 2/20 0.33
P2RX7 Q99572 1/20 0.33
MCHR1 Q99705 1/20 0.33
CYP1A2 P05177 2/20 0.32
CYP2D6 P10635 2/20 0.32
CYP2C9 P11712 2/20 0.32
NPSR1 Q6W5P4 2/20 0.32
MEN1 O00255 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4389111 0.97 LMNA (0.37) PTGES2RETFAAHALDH1A1LMNA
SCHEMBL2008663 0.95 L3MBTL1 (0.36) PTGES2RETFAAHALDH1A1LMNA
SCHEMBL2004824 0.95 PTGES2 (0.36) PTGES2RETFAAHALDH1A1LMNA
SCHEMBL2002979 0.94 LMNA (0.39) PTGES2RETFAAHALDH1A1LMNA
SCHEMBL2001047 0.93 PLA2G2A (0.37) ALDH1A1MAPTKDM4EHPGDCYP1A2
SCHEMBL2003814 0.92 F2RL3 (0.36) PTGES2RETFAAHALDH1A1LMNA
SCHEMBL2006329 0.92 LMNA (0.38) FAAHALDH1A1LMNAMAPTALOX12
SCHEMBL2002134 0.91 PTGES2 (0.42) PTGES2FAAHALDH1A1LMNAMAPT
SCHEMBL2006841 0.91 CYP3A4 (0.37) FAAHALDH1A1LMNAMAPTALOX12
SCHEMBL2009494 0.89 FAAH (0.37) PTGES2FAAHALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed