SCHEMBL2002230

SCHEMBL2002230

Cc1cc(I)cc(Cl)c1N

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CD44 P16070 1/20 0.41
CYP3A4 P08684 4/20 0.40
ALDH1A1 P00352 4/20 0.40
TP53 P04637 1/20 0.40
TSHR P16473 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
CA9 Q16790 2/20 0.35
CYP1A1 P04798 1/20 0.35
CYP1A2 P05177 1/20 0.35
POLB P06746 1/20 0.34
GAA P10253 2/20 0.33
MAPT P10636 1/20 0.33
PLA2G7 Q13093 1/20 0.31
IDO1 P14902 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31729102 1.00 CD44 (0.41) CD44CYP3A4ALDH1A1TP53TSHR
SCHEMBL2861514 0.82 CYP3A4 (0.58) CD44CYP3A4ALDH1A1TP53TSHR
SCHEMBL106150 0.82 ALDH1A1 (0.58) CD44CYP3A4ALDH1A1TP53TSHR
Hydrochloric Acid SCHEMBL27646050 0.79 ALDH1A1 (0.55) CD44CYP3A4ALDH1A1TP53TSHR
Hydrochloric Acid SCHEMBL137754 0.79 ALDH1A1 (0.55) CD44CYP3A4ALDH1A1TP53TSHR
SCHEMBL12834005 0.75 ALDH1A1 (0.43) CD44CYP3A4ALDH1A1TP53TSHR
SCHEMBL1392591 0.75 CYP3A4 (0.65) CD44CYP3A4ALDH1A1TP53TSHR
SCHEMBL698002 0.75 KDM4E (0.45) CD44CYP3A4ALDH1A1TP53TSHR
SCHEMBL18935964 0.75 CA1 (0.52) CYP3A4ALDH1A1TDP1CA1CA2
SCHEMBL30462201 0.75 CD44 (0.44) CD44CYP3A4ALDH1A1TP53TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960584-B2 3-(4-t-butyl-phenyl)-N-(4-methanesulfonylamino-benzyl)-2-methyl-acrylamide; pain, migraine, arthralgia, neuralgia, neuropathies, nerve injury, skin disorder, urinary bladder hypersensitiveness, irritable bowel syndrome, fecal urgency, a respiratory disorder, irritation of skin, eye or mucous membrane AMOREPACIFIC CORPORATION (KR) 2011-06-14 US disclosed
US-20080234383-A1 Novel Compounds, Isomer Thereof, or Pharmaceutically Acceptable Salts Thereof as Vanilloid Receptor Antagonist; and Pharmaceutical Compositions Containing the Same AMOREPACIFIC CORPORATION (KR) 2008-09-25 US disclosed
EP-1861358-A1 NOVEL COMPOUNDS, ISOMER THEREOF, OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF AS VANILLOID RECEPTOR ANTAGONIST, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME Amorepacific Corporation (KR) 2007-12-05 EP disclosed
WO-2006101321-A1 NOVEL COMPOUNDS, ISOMER THEREOF, OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF AS VANILLOID RECEPTOR ANTAGONIST; AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AMOREPACIFIC CORPORATION (KR) 2006-09-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080234383-A1 Novel Compounds, Isomer Thereof, or Pharmaceutically Acceptable Salts Thereof as Vanilloid Receptor Antagonist; and Pharmaceutical Compositions Containing the Same TRPV1, TRPA1, TRPV5 CD44 1749/4885CYP3A4 1203/4885ALDH1A1 612/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.