SCHEMBL2002605

SCHEMBL2002605

Cc1cc2c(C(C)C(=O)O)c(C)n(Cc3cccc(OC(F)(F)F)c3)c2cc1Cl

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 17/20 0.60
PPARA Q07869 11/20 0.60
CYP2C9 P11712 2/20 0.60
EGFR P00533 1/20 0.60
CHRM4 P08173 1/20 0.60
ADRB1 P08588 1/20 0.60
ADRA2A P08913 1/20 0.60
ALOX5 P09917 1/20 0.60
ADRB3 P13945 1/20 0.60
DRD2 P14416 1/20 0.60
ADRA2B P18089 1/20 0.60
CHRM3 P20309 1/20 0.60
TACR2 P21452 1/20 0.60
DRD1 P21728 1/20 0.60
TBXA2R P21731 1/20 0.60
SLC6A2 P23975 1/20 0.60
SLC6A4 P31645 1/20 0.60
OPRM1 P35372 1/20 0.60
PTGER4 P35408 1/20 0.60
DRD3 P35462 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2009343 0.90 PPARG (0.57) PPARGPPARACYP2C9EGFRCHRM4
SCHEMBL3005150 0.85 PPARG (0.57) PPARGPPARACYP2C9EGFRCHRM4
SCHEMBL2006023 0.84 PLA2G2A (0.46) PPARGPPARACYP2C9EGFRCHRM4
SCHEMBL2002573 0.80 PPARG (0.58) PPARGPPARACYP2C9EGFRCHRM4
SCHEMBL2003338 0.79 CCR2 (0.45) PPARGCYP2C9ALOX5CYP1A2CYP2C19
SCHEMBL2001942 0.79 PPARG (0.56) PPARGPPARACYP2C9EGFRCHRM4
SCHEMBL2005057 0.78 PLA2G2A (0.44) PPARGPPARACYP2C9EGFRCHRM4
SCHEMBL2004754 0.77 PPARG (0.56) PPARGPPARACYP2C9EGFRCHRM4
SCHEMBL5547139 0.77 PPARG (0.47) PPARGPPARACYP2C9EGFRCHRM4
SCHEMBL2002879 0.77 PPARG (0.55) PPARGPPARACYP2C9EGFRCHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed
WO-2008103866-A1 SYNTHESIS OF INDOLES MICROBIA, INC. (US) 2008-08-28 WO disclosed