SCHEMBL2002832

SCHEMBL2002832

O=C(c1noc(-c2ccccc2)n1)c1c(C(F)(F)F)n(Cc2ccc(Cl)cc2)c2ccc(O)cc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 2/20 0.40
MAPT P10636 4/20 0.39
PKM P14618 3/20 0.39
GAA P10253 2/20 0.39
ALDH1A1 P00352 1/20 0.39
KDM4E B2RXH2 2/20 0.38
LMNA P02545 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
PTGES2 Q9H7Z7 6/20 0.38
PTGES O14684 2/20 0.38
ABCB11 O95342 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
TBXAS1 P24557 1/20 0.36
HDAC1 Q13547 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
PPARG P37231 1/20 0.35
PLA2G2A P14555 1/20 0.35
TP53 P04637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2009136 0.94 MAPT (0.40) MAPTMEN1KMT2APTGES2PTGES
SCHEMBL2002922 0.92 MAPT (0.35) S1PR3MAPTPKMGAAALDH1A1
SCHEMBL2005007 0.91 PTGES2 (0.40) S1PR3MAPTPKMGAAALDH1A1
SCHEMBL2006486 0.91 PTGES2 (0.41) LMNAMEN1KMT2APTGES2PTGES
SCHEMBL2001735 0.89 MAPT (0.42) S1PR3MAPTPKMGAAALDH1A1
SCHEMBL2004953 0.89 PLA2G2A (0.45) MAPTPKMALDH1A1LMNAMEN1
SCHEMBL2008218 0.87 ALOX5AP (0.41) S1PR3PLA2G2A
SCHEMBL2002572 0.86 HSD17B10 (0.36) S1PR3MAPTALDH1A1KDM4EMEN1
SCHEMBL2004983 0.85 PTGES2 (0.42) MAPTGAAALDH1A1KDM4EMEN1
SCHEMBL2007961 0.85 STAT3 (0.34) S1PR3MAPTPKMGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed