SCHEMBL2002572

SCHEMBL2002572

O=C(c1noc(-c2ccncc2)n1)c1c(C(F)(F)F)n(Cc2ccc(Cl)cc2)c2ccc(Cl)cc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 3/20 0.36
PPARG P37231 3/20 0.36
MAPT P10636 3/20 0.36
CYP3A4 P08684 2/20 0.36
TSHR P16473 2/20 0.36
MEN1 O00255 1/20 0.36
ALOX15 P16050 1/20 0.36
ALOX12 P18054 1/20 0.36
RECQL P46063 1/20 0.36
BLM P54132 1/20 0.36
KMT2A Q03164 1/20 0.36
SRPK1 Q96SB4 1/20 0.35
ALOX5 P09917 1/20 0.34
ALOX5AP P20292 1/20 0.34
STAT3 P40763 1/20 0.34
P2RX3 P56373 1/20 0.34
KDM4E B2RXH2 2/20 0.33
HPGD P15428 2/20 0.33
RHEB Q15382 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2002922 0.94 MAPT (0.35) HSD17B10PPARGMAPTTSHRMEN1
SCHEMBL2006095 0.93 FAAH (0.39) HSD17B10MAPTCYP3A4TSHRMEN1
SCHEMBL2009136 0.92 MAPT (0.40) HSD17B10PPARGMAPTCYP3A4TSHR
SCHEMBL2001648 0.91 RET (0.37) MAPTCYP3A4TSHRALOX12KMT2A
SCHEMBL2006154 0.91 DRD2 (0.37) MAPTCYP3A4MEN1KMT2ASRPK1
SCHEMBL2000833 0.91 KMT2A (0.42) MAPTCYP3A4TSHRMEN1BLM
SCHEMBL2004983 0.90 PTGES2 (0.42) HSD17B10PPARGMAPTCYP3A4TSHR
SCHEMBL2007194 0.90 ALOX5AP (0.42) ALOX5ALOX5APSTAT3S1PR1
SCHEMBL2004742 0.88 STAT3 (0.35) HSD17B10PPARGMAPTCYP3A4TSHR
SCHEMBL2003864 0.88 MAPT (0.38) HSD17B10PPARGMAPTCYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed