SCHEMBL20031661

SCHEMBL20031661

CC(=O)CCCCCOc1ccc2c(c1)CCc1c(C#N)c(C#N)c3c(c1-2)-c1ccccc1CC3

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.42
GLA P06280 1/20 0.42
S1PR1 P21453 2/20 0.39
MAOB P27338 4/20 0.38
MCHR1 Q99705 1/20 0.38
PTPN11 Q06124 1/20 0.38
PDCD1 Q15116 1/20 0.37
CD274 Q9NZQ7 1/20 0.37
EGFR P00533 2/20 0.37
MAPT P10636 2/20 0.36
PDK2 Q15119 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
ALOX12 P18054 1/20 0.36
MAPK1 P28482 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
BRD4 O60885 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22683260 0.86 ITGB3 (0.43) S1PR1MAOBPDK2
SCHEMBL20031890 0.84 MAOB (0.38) KDM4EGLAMAOBEGFRALDH1A1
SCHEMBL22683256 0.83 BRD4 (0.53) KDM4ES1PR1MAOBEGFRMAPT
SCHEMBL20031639 0.81 ALB (0.44) S1PR1MAOBPDK2
SCHEMBL22702989 0.81 THRA (0.47) KDM4EMAOBPTPN11EGFRMAPT
SCHEMBL22683259 0.79 BRD4 (0.48) KDM4ES1PR1MAOBMAPTPDK2
SCHEMBL25017016 0.79 BRD4 (0.57) KDM4EMAOBEGFRMAPTPDK2
SCHEMBL22683275 0.78 ITGB3 (0.38) S1PR1MAOBPDK2
SCHEMBL20031911 0.78 MAOB (0.41) MAOBEGFRMAPK1
SCHEMBL22683261 0.78 MEN1 (0.46) MAOBPTPN11EGFRMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018063105-A1 [5]HELICENE DERIVATIVES AS MOLECULAR REPORTERS FOR DIAGNOSTIC APPLICATIONS AND METHODS OF SYNTHESIS THEREFOR NATIONAL SCIENCE AND TECHNOLOGY DEVELOPMENT AGENCY (TH) 2018-04-05 WO disclosed