SCHEMBL20031900

SCHEMBL20031900

COc1ccc2c(c1)CCc1c(C#N)c(C#N)c3c(c1-2)-c1ccc(OO)cc1CC3

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.53
MAPK1 P28482 1/20 0.48
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
KDM4E B2RXH2 4/20 0.43
GLA P06280 3/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 2/20 0.42
TP53 P04637 1/20 0.42
POLB P06746 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
ALPL P05186 1/20 0.42
CLK1 P49759 1/20 0.42
HSD17B10 Q99714 1/20 0.42
RAB9A P51151 2/20 0.40
ATM Q13315 2/20 0.40
NPC1 O15118 1/20 0.40
MAP3K9 P80192 1/20 0.39
MAP3K11 Q16584 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22703046 0.93 EGFR (0.44) EGFRMAPK1CYP1A2CYP2D6KDM4E
SCHEMBL20031646 0.93 EGFR (0.58) EGFRMAPK1CYP1A2CYP2D6KDM4E
SCHEMBL25016883 0.87 EGFR (0.42) EGFRMAPK1NOTUMCYP26A1MIF
SCHEMBL20031875 0.85 EGFR (0.51) EGFRMAPK1CYP1A2CYP2D6KDM4E
SCHEMBL20031910 0.78 EGFR (0.44) EGFRMAPK1KDM4EGLAALDH1A1
SCHEMBL20031643 0.78 MAPK1 (0.42) EGFRMAPK1CYP1A2ALDH1A1MEN1
SCHEMBL20031659 0.74 MIF (0.44) EGFRMAPK1CYP1A2KDM4EALDH1A1
SCHEMBL22702989 0.73 THRA (0.47) EGFRKDM4EALDH1A1MAPTMEN1
SCHEMBL7284412 0.71 BCL2 (0.49) EGFRMAPK1CYP1A2CYP2D6KDM4E
SCHEMBL22683261 0.71 MEN1 (0.46) EGFRALDH1A1MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018063105-A1 [5]HELICENE DERIVATIVES AS MOLECULAR REPORTERS FOR DIAGNOSTIC APPLICATIONS AND METHODS OF SYNTHESIS THEREFOR NATIONAL SCIENCE AND TECHNOLOGY DEVELOPMENT AGENCY (TH) 2018-04-05 WO disclosed