SCHEMBL2003255

SCHEMBL2003255

CCOc1ccc2c(c1)c(C(=O)c1nc(-c3ccncc3)no1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
LMNA P02545 3/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
HPGD P15428 2/20 0.38
TP53 P04637 2/20 0.38
TSHR P16473 1/20 0.38
NFKB1 P19838 1/20 0.38
CASP3 P42574 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
SENP8 Q96LD8 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
SENP6 Q9GZR1 1/20 0.38
S1PR1 P21453 3/20 0.37
MAPT P10636 3/20 0.36
GSTP1 P09211 1/20 0.36
F2RL3 Q96RI0 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
SMPD1 P17405 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2007930 0.94 PLA2G2A (0.38) NPC1RAB9ALMNASMN1; SMN2HPGD
SCHEMBL2002951 0.92 S1PR1 (0.41) NPC1RAB9ALMNASMN1; SMN2TP53
SCHEMBL2001517 0.91 ALOX5AP (0.42) NPC1RAB9ALMNASMN1; SMN2TSHR
SCHEMBL2003332 0.91 SMN1; SMN2 (0.39) NPC1RAB9ALMNASMN1; SMN2HPGD
SCHEMBL2002732 0.91 LMNA (0.33) LMNASMN1; SMN2MAPTF2RL3F10
SCHEMBL2001583 0.90 LMNA (0.40) NPC1RAB9ALMNASMN1; SMN2HPGD
SCHEMBL2007825 0.89 TP53 (0.43) NPC1RAB9ALMNASMN1; SMN2HPGD
SCHEMBL2002547 0.88 RAB9A (0.39) NPC1RAB9ALMNASMN1; SMN2HPGD
SCHEMBL2003150 0.88 S1PR1 (0.35) LMNASMN1; SMN2HPGDS1PR1MAPT
SCHEMBL2008151 0.88 LMNA (0.39) NPC1RAB9ALMNASMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed