SCHEMBL20032577

SCHEMBL20032577

CC(=O)[C@H]1C[C@@H]1C(=O)c1cc(Cl)c2c(c1)CC(C)O2

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KMO O15229 2/20 0.39
PARP1 P09874 6/20 0.39
TDP1 Q9NUW8 1/20 0.38
AKR1B1 P15121 7/20 0.33
MAOA P21397 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16600346 0.90 KMO (0.51) KMOPARP1TDP1AKR1B1
SCHEMBL16600309 0.90 KMO (0.51) KMOPARP1TDP1AKR1B1
SCHEMBL21218966 0.90 KMO (0.51) KMOPARP1TDP1AKR1B1
SCHEMBL21231297 0.90 KMO (0.51) KMOPARP1TDP1AKR1B1
SCHEMBL16614134 0.88 KMO (0.37) KMOPARP1TDP1AKR1B1MAOA
SCHEMBL20032572 0.85 KMO (0.37) KMO
SCHEMBL20032576 0.78 KMO (0.40) KMOAKR1B1
SCHEMBL20032573 0.76 TDP1 (0.63) KMOTDP1AKR1B1MAOA
SCHEMBL21231402 0.75 KMO (0.49) KMOTDP1AKR1B1
SCHEMBL16614133 0.75 KMO (0.49) KMOTDP1AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9938252-B2 Kynurenine-3-monooxygenase inhibitors, pharmaceutical compositions, and methods of use thereof CHDI FOUNDATION, INC. (US) 2018-04-10 US disclosed