SCHEMBL2004267

SCHEMBL2004267

CCOc1ccc2c(c1)c(C(=O)c1noc(-c3cccnc3)n1)c(Cl)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 2/20 0.42
NPC1 O15118 5/20 0.41
SMN1; SMN2 Q16637 5/20 0.41
RAB9A P51151 4/20 0.41
TP53 P04637 3/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
MAPT P10636 7/20 0.37
LMNA P02545 4/20 0.37
KMT2A Q03164 1/20 0.37
PKM P14618 1/20 0.37
CYP19A1 P11511 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
ALOX5AP P20292 3/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2002749 0.93 NPC1 (0.41) NPC1SMN1; SMN2RAB9ATP53MAPT
SCHEMBL2003533 0.92 S1PR1 (0.44) S1PR1NPC1SMN1; SMN2RAB9ATP53
SCHEMBL2007918 0.92 ALOX5AP (0.40) S1PR1SMN1; SMN2MAPTLMNAALOX5AP
SCHEMBL2005122 0.91 S1PR1 (0.38) S1PR1SMN1; SMN2MAPTLMNAALOX5AP
SCHEMBL2007600 0.91 S1PR1 (0.40) S1PR1NPC1SMN1; SMN2RAB9ATP53
SCHEMBL2006916 0.91 LMNA (0.37) NPC1SMN1; SMN2RAB9ATP53MAPT
SCHEMBL2004109 0.89 LMNA (0.36) NPC1SMN1; SMN2RAB9ATP53NFKB1
SCHEMBL2006526 0.88 L3MBTL1 (0.39) NPC1RAB9AMAPTLMNAPKM
SCHEMBL2009470 0.88 S1PR1 (0.43) S1PR1NPC1SMN1; SMN2RAB9ATP53
SCHEMBL2006172 0.87 ALOX5AP (0.39) SMN1; SMN2MAPTLMNAKMT2ACYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed