SCHEMBL2003154

SCHEMBL2003154

CCOc1ccc2c(c1)c(C(=O)c1noc(-c3ccccc3)n1)c(Cl)n2Cc1ccc(Cl)cc1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 2/20 0.42
S1PR1 P21453 1/20 0.42
S1PR5 Q9H228 1/20 0.42
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
PLA2G2A P14555 2/20 0.40
ALOX5 P09917 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NTRK1 P04629 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2003734 0.93 ALOX5AP (0.42) ALOX5APS1PR1S1PR5PTGS1PTGS2
SCHEMBL2001661 0.92 PLA2G2A (0.48) PTGS2PLA2G2AMAPTKMT2A
SCHEMBL2003533 0.91 S1PR1 (0.44) ALOX5APS1PR1ALOX5MAPTKMT2A
SCHEMBL2007918 0.91 ALOX5AP (0.40) ALOX5APS1PR1S1PR5MAPTSMN1; SMN2
SCHEMBL2008218 0.90 ALOX5AP (0.41) ALOX5APS1PR1S1PR5PTGS1PTGS2
SCHEMBL2003080 0.90 ALOX5AP (0.41) ALOX5APPTGS1PTGS2ALOX5MAPT
SCHEMBL1999518 0.89 MAPT (0.43) S1PR1S1PR5MAPTKMT2A
SCHEMBL2003586 0.87 KMT2A (0.42) ALOX5MAPTKMT2ASMN1; SMN2
SCHEMBL2001735 0.86 MAPT (0.42) S1PR1S1PR5PLA2G2AMAPTKMT2A
SCHEMBL2011061 0.85 ALOX5AP (0.39) ALOX5APPTGS1PTGS2ALOX5MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed