SCHEMBL20042735

SCHEMBL20042735

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)C1CCC(F)(F)CC1)C2

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 3/20 0.41
CNR1 P21554 2/20 0.39
GPR55 Q9Y2T6 2/20 0.39
GRM5 P41594 4/20 0.38
CHRM4 P08173 1/20 0.36
LMNA P02545 1/20 0.35
TSHR P16473 1/20 0.35
NR4A1 P22736 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PIK3CD O00329 1/20 0.34
PIK3CA P42336 1/20 0.34
SCN10A Q9Y5Y9 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GBA1 P04062 1/20 0.32
GPR6 P46095 2/20 0.32
NAMPT P43490 1/20 0.32
HSD11B1 P28845 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042785 0.94 CNR2 (0.36) CNR2CNR1GPR55GRM5CHRM4
SCHEMBL20042779 0.90 GPR55 (0.39) CNR2CNR1GPR55CHRM4LMNA
SCHEMBL20042806 0.88 CNR1 (0.47) CNR1GPR55CHRM4LMNATSHR
SCHEMBL20042800 0.88 CNR1 (0.45) CNR1GPR55CHRM4LMNATSHR
SCHEMBL20042764 0.87 CNR1 (0.49) CNR1GPR55LMNATSHRNR4A1
SCHEMBL20042816 0.85 CNR1 (0.45) CNR2CNR1GPR55GRM5CHRM4
SCHEMBL20042706 0.84 ALDH1A1 (0.43) CNR2CNR1GPR55CHRM4LMNA
SCHEMBL20042762 0.83 CNR1 (0.40) CNR2CNR1GPR55GRM5LMNA
SCHEMBL20042793 0.83 SMN1; SMN2 (0.37) CNR1GPR55GRM5CHRM4LMNA
SCHEMBL20042660 0.81 CNR1 (0.39) CNR2CNR1GPR55GRM5LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed