SCHEMBL20042865

SCHEMBL20042865

Cc1nc2c(c(N3CCC3)n1)C(C)N(C(=O)c1ccc(F)cc1)C2

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 19/20 0.42
CYP2C9 P11712 4/20 0.42
CYP2C19 P33261 4/20 0.42
CYP1A2 P05177 2/20 0.42
KCNH2 Q12809 4/20 0.42
CYP3A4 P08684 2/20 0.42
TACR2 P21452 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042958 1.00 TACR3 (0.42) TACR3CYP2C9CYP2C19CYP1A2KCNH2
SCHEMBL20042982 0.89 P2RX7 (0.46) TACR3CYP2C9CYP2C19CYP1A2KCNH2
SCHEMBL20042851 0.89 P2RX7 (0.46) TACR3CYP2C9CYP2C19CYP1A2KCNH2
SCHEMBL20042900 0.88 TACR3 (0.38) TACR3KCNH2TACR2
SCHEMBL20042898 0.88 TACR3 (0.45) TACR3CYP2C9CYP2C19CYP1A2KCNH2
SCHEMBL20042767 0.86 TACR3 (0.44) TACR3KCNH2
SCHEMBL20042928 0.86 TACR3 (0.44) TACR3CYP2C9CYP2C19CYP1A2KCNH2
SCHEMBL20042727 0.86 TACR3 (0.47) TACR3KCNH2TACR2
SCHEMBL20042852 0.86 TACR3 (0.47) TACR3KCNH2TACR2
SCHEMBL20042878 0.86 TACR3 (0.47) TACR3KCNH2TACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed