SCHEMBL20042834

SCHEMBL20042834

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)CC1CC1)C2

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 14/20 0.56
CYP1A2 P05177 2/20 0.56
ADORA2A P29274 1/20 0.46
ADORA1 P30542 1/20 0.46
CHRM2 P08172 4/20 0.38
LMNA P02545 1/20 0.35
TSHR P16473 1/20 0.35
NR4A1 P22736 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NAMPT P43490 1/20 0.35
CNR2 P34972 1/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CNR1 P21554 1/20 0.33
GPR55 Q9Y2T6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042651 0.96 CHRM4 (0.52) CHRM4CYP1A2ADORA2AADORA1CHRM2
SCHEMBL20042773 0.96 CHRM4 (0.52) CHRM4CYP1A2ADORA2AADORA1CHRM2
SCHEMBL20042714 0.88 CHRM4 (0.43) CHRM4CYP1A2ADORA2AADORA1LMNA
SCHEMBL20042654 0.85 HSD11B1 (0.41) CHRM4CYP1A2ADORA2AADORA1LMNA
SCHEMBL20042806 0.80 CNR1 (0.47) CHRM4LMNATSHRNR4A1SMN1; SMN2
SCHEMBL20042800 0.80 CNR1 (0.45) CHRM4CYP1A2LMNATSHRNR4A1
SCHEMBL31614812 0.80 CHRM4 (0.70) CHRM4CYP1A2CHRM2
SCHEMBL31614814 0.80 CHRM4 (0.70) CHRM4CYP1A2CHRM2
SCHEMBL20042870 0.79 KDM4E (0.35) LMNATSHRNR4A1SMN1; SMN2KDM4E
SCHEMBL20042764 0.79 CNR1 (0.49) LMNATSHRNR4A1SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed