SCHEMBL20042654

SCHEMBL20042654

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)CCC1CCCC1)C2

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.41
ALDH1A1 P00352 8/20 0.41
ATM Q13315 2/20 0.41
TP53 P04637 1/20 0.40
KMT2A Q03164 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CHRM4 P08173 1/20 0.40
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39
CNR2 P34972 3/20 0.38
LMNA P02545 2/20 0.38
CNR1 P21554 1/20 0.38
KDM4E B2RXH2 1/20 0.37
MAPT P10636 1/20 0.37
HIF1A Q16665 1/20 0.37
MEN1 O00255 1/20 0.37
LDHA P00338 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042714 0.97 CHRM4 (0.43) HSD11B1ALDH1A1ATMTP53KMT2A
SCHEMBL20042651 0.88 CHRM4 (0.52) ALDH1A1SMN1; SMN2CYP1A2CHRM4ADORA2A
SCHEMBL20042773 0.86 CHRM4 (0.52) ALDH1A1SMN1; SMN2CYP1A2CHRM4ADORA2A
SCHEMBL20042834 0.85 CHRM4 (0.56) ALDH1A1SMN1; SMN2CYP1A2CHRM4ADORA2A
SCHEMBL20042650 0.80 USP19 (0.37) CYP1A2CHRM4ADORA2AADORA1CNR1
SCHEMBL20042806 0.80 CNR1 (0.47) HSD11B1ALDH1A1KMT2ASMN1; SMN2CHRM4
SCHEMBL20042764 0.79 CNR1 (0.49) HSD11B1ALDH1A1KMT2ASMN1; SMN2LMNA
SCHEMBL20042748 0.78 NPC1 (0.49) ALDH1A1KMT2ASMN1; SMN2MAPTMEN1
SCHEMBL20042690 0.77 GFER (0.41) ALDH1A1KMT2ACHRM4LMNAMEN1
SCHEMBL20042830 0.76 ME2 (0.43) ALDH1A1KMT2AMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed