SCHEMBL20042773

SCHEMBL20042773

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)CC1CCC1)C2

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 14/20 0.52
CYP1A2 P05177 2/20 0.52
ADORA2A P29274 1/20 0.47
ADORA1 P30542 1/20 0.47
CHRM2 P08172 4/20 0.37
CNR2 P34972 2/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HSD17B10 Q99714 1/20 0.35
LMNA P02545 1/20 0.35
TSHR P16473 1/20 0.35
NR4A1 P22736 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPY5R Q15761 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042651 0.98 CHRM4 (0.52) CHRM4CYP1A2ADORA2AADORA1CHRM2
SCHEMBL20042834 0.96 CHRM4 (0.56) CHRM4CYP1A2ADORA2AADORA1CHRM2
SCHEMBL20042654 0.86 HSD11B1 (0.41) CHRM4CYP1A2ADORA2AADORA1CNR2
SCHEMBL20042714 0.85 CHRM4 (0.43) CHRM4CYP1A2ADORA2AADORA1CNR2
SCHEMBL20042800 0.81 CNR1 (0.45) CHRM4CYP1A2ALDH1A1LMNATSHR
SCHEMBL20042650 0.80 USP19 (0.37) CHRM4CYP1A2ADORA2AADORA1NPY5R
SCHEMBL20042806 0.79 CNR1 (0.47) CHRM4ALDH1A1LMNATSHRNR4A1
SCHEMBL31614812 0.79 CHRM4 (0.70) CHRM4CYP1A2CHRM2
SCHEMBL31614814 0.79 CHRM4 (0.70) CHRM4CYP1A2CHRM2
SCHEMBL20042870 0.78 KDM4E (0.35) KDM4EALDH1A1HSD17B10LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed