SCHEMBL20042898

SCHEMBL20042898

Cc1nc2c(c(N3CCC3)n1)[C@@H](C)N(C(=O)c1cccc(F)c1)C2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 1/20 0.45
KCNH2 Q12809 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
PIK3CD O00329 1/20 0.41
KDM4E B2RXH2 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
GRM5 P41594 4/20 0.41
ALDH1A1 P00352 2/20 0.39
HPGD P15428 1/20 0.39
USP2 O75604 2/20 0.39
LMNA P02545 1/20 0.39
NPY5R Q15761 1/20 0.38
RAB9A P51151 1/20 0.37
P2RX7 Q99572 1/20 0.37
ABL1 P00519 1/20 0.37
BCR P11274 1/20 0.37
CYP3A4 P08684 1/20 0.37
MAPT P10636 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042841 0.88 TACR2 (0.45) TACR3KCNH2KDM4ETDP1GRM5
SCHEMBL20042958 0.88 TACR3 (0.42) TACR3KCNH2CYP3A4CYP1A2CYP2C9
SCHEMBL20042865 0.88 TACR3 (0.42) TACR3KCNH2CYP3A4CYP1A2CYP2C9
SCHEMBL20042989 0.87 SMN1; SMN2 (0.44) TACR3KCNH2SMN1; SMN2PIK3CDKDM4E
SCHEMBL20042991 0.87 SMN1; SMN2 (0.41) TACR3KCNH2SMN1; SMN2PIK3CDKDM4E
SCHEMBL20042900 0.86 TACR3 (0.38) TACR3KCNH2ALDH1A1P2RX7
SCHEMBL20042894 0.85 GRM5 (0.40) GRM5P2RX7
SCHEMBL20042843 0.85 GRM5 (0.40) GRM5P2RX7
SCHEMBL20042986 0.85 TAS1R3 (0.40) TACR3KCNH2TDP1GRM5LMNA
SCHEMBL20042876 0.85 TAS1R3 (0.40) TACR3KCNH2TDP1GRM5LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed