SCHEMBL20042841

SCHEMBL20042841

Cc1nc2c(c(N3CCC3)n1)C(C)N(C(=O)c1cccc(Cl)c1)C2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 1/20 0.45
TACR3 P29371 1/20 0.45
KCNH2 Q12809 1/20 0.45
LMNA P02545 2/20 0.42
PARP1 P09874 1/20 0.39
ALDH1A1 P00352 4/20 0.39
PKM P14618 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
PGR P06401 1/20 0.39
KMT2A Q03164 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
HSP90AA1 P07900 1/20 0.38
MAPT P10636 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
KDM2B Q8NHM5 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042898 0.88 TACR3 (0.45) TACR3KCNH2LMNAALDH1A1KDM4E
SCHEMBL20042851 0.88 P2RX7 (0.46) TACR2TACR3KCNH2LMNAALDH1A1
SCHEMBL20042982 0.88 P2RX7 (0.46) TACR2TACR3KCNH2LMNAALDH1A1
SCHEMBL20042922 0.87 TACR2 (0.40) TACR2TACR3KCNH2LMNAALDH1A1
SCHEMBL20042927 0.87 TACR2 (0.40) TACR2TACR3KCNH2LMNAALDH1A1
SCHEMBL20042868 0.87 P2RX7 (0.35) TACR2TACR3KCNH2LMNAKMT2A
SCHEMBL20042852 0.86 TACR3 (0.47) TACR2TACR3KCNH2
SCHEMBL20042883 0.86 GPR6 (0.39) TACR2TACR3KCNH2LMNAKDM4E
SCHEMBL20042983 0.86 GPR6 (0.39) TACR2TACR3KCNH2LMNAKDM4E
SCHEMBL20042843 0.85 GRM5 (0.40) GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed